SCHEMBL22967337

SCHEMBL22967337

Nc1nc2[nH]cc(CCc3ccccc3)c2c(=O)[nH]1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TYMS P04818 10/20 0.59
FOLR1 P15328 2/20 0.59
SLC19A1 P41440 2/20 0.59
SLC46A1 Q96NT5 2/20 0.59
DHFR P00374 1/20 0.59
FOLR2 P14207 1/20 0.59
GART P22102 1/20 0.59
ATIC P31939 1/20 0.59
SHMT1 P34896 1/20 0.59
FRK P42685 1/20 0.59
PNP P00491 1/20 0.52
BACE1 P56817 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12238856 0.87 TYMS (0.57) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL29094260 0.86 TYMS (0.50) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL2260428 0.86 TYMS (0.69) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL2260030 0.85 TYMS (0.67) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL18755599 0.85 TYMS (0.55) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL17652074 0.84 TYMS (0.48) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL24845712 0.84 TYMS (0.56) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL18551642 0.84 TYMS (0.64) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL30130170 0.84 TYMS (0.66) TYMSFOLR1SLC19A1SLC46A1DHFR
SCHEMBL24845716 0.84 PNP (0.57) TYMSFOLR1SLC19A1SLC46A1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021026310-A1 PROCESSES OF PREPARING POLYGLUTAMATED ANTIFOLATES AND USES OF THEIR COMPOSITIONS L.E.A.F. HOLDINGS GROUP LLC (US) 2021-02-11 WO disclosed