SCHEMBL22969844

SCHEMBL22969844

C=BN1CCc2c(nc(Cl)nc2N2CCN(C(=O)OC(C)(C)C)C(CC#N)C2)C1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.40
VHL P40337 1/20 0.39
CDK7 P50613 1/20 0.39
CCNH P51946 1/20 0.39
MNAT1 P51948 1/20 0.39
SOS1 Q07889 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27230441 0.87 KRAS (0.40) KRASVHLCDK7CCNHMNAT1
SCHEMBL29039717 0.87 KRAS (0.40) KRASVHLCDK7CCNHMNAT1
SCHEMBL27210008 0.87 KRAS (0.40) KRASVHLCDK7CCNHMNAT1
SCHEMBL19617686 0.83 KRAS (0.42) KRASVHLCDK7CCNHMNAT1
SCHEMBL19637829 0.83 KRAS (0.42) KRASVHLCDK7CCNHMNAT1
SCHEMBL29493372 0.83 KRAS (0.42) KRASVHLCDK7CCNHMNAT1
SCHEMBL23074825 0.81 PARP1 (0.39) KRASVHLCDK7CCNHMNAT1
SCHEMBL19948615 0.81 PARP1 (0.46) KRASVHLCDK7CCNHMNAT1
SCHEMBL24528933 0.81 KRAS (0.61) KRASVHLCDK7CCNHMNAT1
SCHEMBL23075034 0.80 NR1H2 (0.42) KRASVHLCDK7CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021023247-A1 KRAS MUTANT PROTEIN INHIBITOR JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2021-02-11 WO disclosed