SCHEMBL29039717

SCHEMBL29039717

CC(C)(C)OC(=O)N1CCN(c2nc(Cl)nc3c2CCN(C(=O)O)C3)C[C@H]1CC#N

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KRAS P01116 18/20 0.40
VHL P40337 1/20 0.39
CDK7 P50613 1/20 0.39
CCNH P51946 1/20 0.39
MNAT1 P51948 1/20 0.39
SOS1 Q07889 1/20 0.39
MTOR P42345 1/20 0.37
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27230441 1.00 KRAS (0.40) KRASVHLCDK7CCNHMNAT1
SCHEMBL27210008 1.00 KRAS (0.40) KRASVHLCDK7CCNHMNAT1
SCHEMBL21315017 0.89 KRAS (0.37) KRASVHLCDK7CCNHMNAT1
SCHEMBL21315015 0.89 KRAS (0.37) KRASVHLCDK7CCNHMNAT1
SCHEMBL23827647 0.88 MTOR (0.37) KRASVHLCDK7CCNHMNAT1
SCHEMBL28504722 0.88 MTOR (0.38) KRASMTORNR1H2NR1H3
SCHEMBL19948615 0.88 PARP1 (0.46) KRASVHLCDK7CCNHMNAT1
SCHEMBL22969844 0.87 KRAS (0.40) KRASVHLCDK7CCNHMNAT1
SCHEMBL19948470 0.87 MTOR (0.37) KRASMTORNR1H2NR1H3
SCHEMBL19948468 0.87 MTOR (0.37) KRASMTORNR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478184-A KRAS inhibitor and preparation method and application thereof 上海华汇拓医药科技有限公司 2023-07-25 CN disclosed