SCHEMBL2297279

SCHEMBL2297279

COc1cc(C(=O)NC2CCN(C(=O)O)CC2)ccc1Nc1ncc2c(n1)N(C1CCCCC1)CC(F)(F)C(=O)N2C

nearest known ligand 0.87

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 18/20 0.87
BRD4 O60885 5/20 0.87
BRDT Q58F21 5/20 0.87
RAD52 P43351 1/20 0.68
ALK Q9UM73 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2299916 0.99 PLK1 (0.88) PLK1BRD4BRDTRAD52ALK
SCHEMBL12330693 0.94 PLK1 (0.92) PLK1BRD4BRDTRAD52ALK
SCHEMBL1559612 0.94 PLK1 (0.92) PLK1BRD4BRDTRAD52ALK
SCHEMBL2298489 0.94 PLK1 (0.79) PLK1BRD4BRDTRAD52ALK
SCHEMBL1675705 0.94 PLK1 (0.88) PLK1BRD4BRDTRAD52ALK
SCHEMBL1560010 0.94 PLK1 (0.99) PLK1BRD4BRDTRAD52ALK
SCHEMBL1675854 0.94 PLK1 (0.90) PLK1BRD4BRDTRAD52ALK
SCHEMBL2299733 0.93 PLK1 (0.82) PLK1BRD4BRDTRAD52
SCHEMBL1559146 0.93 PLK1 (1.00) PLK1BRD4BRDTRAD52ALK
SCHEMBL29377237 0.93 PLK1 (1.00) PLK1BRD4BRDTRAD52ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003785-B2 Halo-substituted pyrimidodiazepines TAKEDA PHARMACEUTICAL COMPANY LIMITED (US) 2011-08-23 US disclosed