SCHEMBL2298489

SCHEMBL2298489

CCOc1cc(C(=O)NC2CCN(C(=O)O)CC2)ccc1Nc1ncc2c(n1)N(C1CCCC1)CC(F)(F)C(=O)N2C

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 16/20 0.79
BRD4 O60885 4/20 0.79
BRDT Q58F21 3/20 0.79
ALK Q9UM73 3/20 0.71
RAD52 P43351 1/20 0.60
PLK3 Q9H4B4 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2299916 0.95 PLK1 (0.88) PLK1BRD4BRDTALKRAD52
SCHEMBL2297279 0.94 PLK1 (0.87) PLK1BRD4BRDTALKRAD52
SCHEMBL1560504 0.94 PLK1 (0.90) PLK1BRD4BRDTALKRAD52
SCHEMBL1559962 0.93 PLK1 (0.80) PLK1BRD4BRDTALKRAD52
SCHEMBL2299520 0.92 PLK1 (0.73) PLK1BRD4BRDTALKRAD52
SCHEMBL1559955 0.92 PLK1 (0.75) PLK1BRD4BRDTALKRAD52
SCHEMBL1559565 0.91 PLK1 (0.74) PLK1BRD4BRDTALKRAD52
SCHEMBL1559954 0.91 PLK1 (0.77) PLK1BRD4BRDTALKRAD52
SCHEMBL1560365 0.91 PLK1 (0.77) PLK1BRD4BRDTALKRAD52
SCHEMBL2299583 0.91 PLK1 (0.74) PLK1BRD4BRDTALKRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003785-B2 Halo-substituted pyrimidodiazepines TAKEDA PHARMACEUTICAL COMPANY LIMITED (US) 2011-08-23 US disclosed