SCHEMBL2298218

SCHEMBL2298218

CNC(=O)c1c(-c2ccccc2)oc2cc(NS(C)(=O)=O)c(C3CC3)cc12

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.48
CYP3A4 P08684 5/20 0.48
CYP2C19 P33261 4/20 0.48
KCNH2 Q12809 3/20 0.48
TP53 P04637 2/20 0.38
MAPT P10636 2/20 0.38
CYP2C8 P10632 1/20 0.37
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2294325 0.90 CYP2C9 (0.53) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2298808 0.90 CYP2C9 (0.59) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6119827 0.90 CYP2C9 (0.51) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6119825 0.88 CYP2C9 (0.49) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6119471 0.87 CYP2C9 (0.51) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2300601 0.85 CYP2C9 (0.54) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2296799 0.82 CYP2C9 (0.43) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2295568 0.82 CYP2C9 (0.48) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6119844 0.82 CYP2C9 (0.50) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6120266 0.82 CYP2C9 (0.41) CYP2C9CYP3A4CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103063-A1 THERAPEUTIC COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-08-25 WO disclosed