SCHEMBL2298467

SCHEMBL2298467

CS(=O)(=O)Nc1cc2oc(-c3ccc(F)cc3)c(C(N)=O)c2cc1C1CC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2C19 P33261 4/20 0.47
KCNH2 Q12809 2/20 0.47
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
ANO1 Q5XXA6 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6119722 0.96 CYP2C9 (0.45) CYP2C9CYP3A4CYP2C19KCNH2RAB9A
SCHEMBL2295568 0.91 CYP2C9 (0.48) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL2298808 0.89 CYP2C9 (0.59) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6119844 0.89 CYP2C9 (0.50) CYP2C9CYP3A4CYP2C19KCNH2RAB9A
SCHEMBL6119377 0.87 CYP2C9 (0.49) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2298813 0.87 CYP2C9 (0.50) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL9952934 0.86 CYP2C9 (0.46) CYP2C9CYP3A4CYP2C19KCNH2KDM4E
SCHEMBL4758844 0.86 CYP2C9 (0.48) CYP2C9CYP3A4CYP2C19KCNH2KDM4E
SCHEMBL2302690 0.86 CYP2C9 (0.45) CYP2C9CYP3A4CYP2C19KCNH2KDM4E
SCHEMBL2300601 0.85 CYP2C9 (0.54) CYP2C9CYP3A4CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012067663-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-05-24 WO disclosed
WO-2011103063-A1 THERAPEUTIC COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-08-25 WO disclosed