SCHEMBL2298687

SCHEMBL2298687

CCOC(=O)C(F)(F)CN(c1nc(Cl)ncc1[N+](=O)[O-])C1CC1c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 13/20 0.37
MAPT P10636 4/20 0.34
LMNA P02545 3/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CES2 O00748 1/20 0.33
ACHE P22303 1/20 0.33
CES1 P23141 1/20 0.33
DHFR P00374 1/20 0.33
ALOX12 P18054 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2298690 1.00 PIN1 (0.37) PIN1MAPTLMNAALDH1A1SMN1; SMN2
SCHEMBL29259965 0.83 PIN1 (0.34) PIN1MAPTLMNAALDH1A1NPSR1
SCHEMBL30938311 0.83 PIN1 (0.34) PIN1MAPTLMNAALDH1A1NPSR1
SCHEMBL2302176 0.83 MEN1 (0.34) PIN1MAPTLMNAALDH1A1NPSR1
SCHEMBL1675935 0.82 MEN1 (0.35) PIN1MAPTLMNAALDH1A1SMN1; SMN2
SCHEMBL1560434 0.81 KMT2A (0.37) PIN1MAPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL1675637 0.81 PIN1 (0.32) PIN1
SCHEMBL2300832 0.78 PIN1 (0.46) PIN1MAPTLMNAALDH1A1CES2
SCHEMBL30965570 0.78 PIN1 (0.36) PIN1MAPTLMNAALDH1A1NPSR1
SCHEMBL2295524 0.77 PIN1 (0.45) PIN1MAPTLMNASMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003785-B2 Halo-substituted pyrimidodiazepines TAKEDA PHARMACEUTICAL COMPANY LIMITED (US) 2011-08-23 US disclosed
US-20090318408-A1 HALO-SUBSTITUTED PYRIMIDODIAZEPINES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318408-A1 HALO-SUBSTITUTED PYRIMIDODIAZEPINES PLK1, CCNI, CDK1 PIN1 292/4885MAPT 2512/4885LMNA 2080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.