SCHEMBL22987598

SCHEMBL22987598

CSc1ccccc1-c1nc2c3ccccc3[nH]c(=O)n2n1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 1/20 0.63
GABRD O14764 1/20 0.63
GABRA1 P14867 1/20 0.63
GABRB1 P18505 1/20 0.63
GABRG2 P18507 1/20 0.63
GABRB3 P28472 1/20 0.63
GABRA5 P31644 1/20 0.63
GABRA3 P34903 1/20 0.63
GABRA2 P47869 1/20 0.63
GABRB2 P47870 1/20 0.63
GABRA4 P48169 1/20 0.63
GABRE P78334 1/20 0.63
GABRA6 Q16445 1/20 0.63
GABRG1 Q8N1C3 1/20 0.63
GABRG3 Q99928 1/20 0.63
GABRQ Q9UN88 1/20 0.63
TP53 P04637 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
RXFP1 Q9HBX9 1/20 0.61
HAVCR2 Q8TDQ0 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979071 0.84 TP53 (0.69) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29646306 0.84 TP53 (0.69) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22987516 0.81 TP53 (0.77) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL10715371 0.81 GABRP (0.67) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22988165 0.81 GABRP (0.67) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29646362 0.81 GABRP (0.67) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22979964 0.81 GABRP (0.67) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29646443 0.81 GABRP (0.67) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22987597 0.81 GABRP (0.63) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22979237 0.81 KDM4E (0.67) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021028382-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed