SCHEMBL22987915

SCHEMBL22987915

Nc1nc2ccccc2c2nc(-c3ccc(OC(F)(F)F)cc3)nn12

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 12/20 0.50
ADORA1 P30542 4/20 0.50
ADORA2A P29274 6/20 0.48
ACP1 P24666 1/20 0.45
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
NOD1 Q9Y239 1/20 0.44
ADA P00813 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22988327 0.87 ADORA1 (0.47) ADORA3ADORA1ADORA2AACP1MAPT
SCHEMBL22979755 0.86 ADORA3 (0.50) ADORA3ADORA1ADORA2AACP1MAPT
SCHEMBL29646450 0.86 ADORA3 (0.50) ADORA3ADORA1ADORA2AACP1MAPT
SCHEMBL22988304 0.84 ADORA3 (0.65) ADORA3ADORA1ADORA2AMAPTTHRB
SCHEMBL22987511 0.82 ADORA3 (0.45) ADORA3ADORA1ADORA2AMAPTADA
SCHEMBL31150001 0.80 ADORA3 (0.41) ADORA3ADORA1ADORA2AACP1MAPT
SCHEMBL22988235 0.78 ADORA3 (0.51) ADORA3ADORA1ADORA2AMAPT
SCHEMBL30393303 0.77 NPC1 (0.52) ADORA3ADORA1ADORA2AACP1MAPT
SCHEMBL22988309 0.77 ADORA3 (0.53) ADORA3ADORA1ADORA2AMAPT
SCHEMBL22988361 0.76 PDE10A (0.53) ADORA3ADORA1ADORA2AMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021028382-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed