SCHEMBL23002201

SCHEMBL23002201

Cc1ccc(F)c(C2(NC(=O)OC(C)(C)C)CCCCC2=O)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 3/20 0.35
GRIN1 Q05586 3/20 0.34
GRIN2A Q12879 3/20 0.34
HDAC4 P56524 3/20 0.34
GRIN2B Q13224 2/20 0.34
PPIA P62937 2/20 0.34
SLC6A4 P31645 2/20 0.33
OPRK1 P41145 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
LMNA P02545 1/20 0.33
OPRM1 P35372 1/20 0.33
CACNA1C Q13936 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452505 0.89 GRIN1 (0.38) BDKRB1GRIN1GRIN2AGRIN2BSLC6A4
SCHEMBL21452562 0.85 KCNQ3 (0.37) GRIN1GRIN2AGRIN2BPPIASLC6A4
SCHEMBL21451917 0.83 GRIN1 (0.40) BDKRB1GRIN1GRIN2AGRIN2BSLC6A4
SCHEMBL23002199 0.83 BDKRB1 (0.34) BDKRB1OPRK1LMNA
SCHEMBL21452415 0.81 HDAC4 (0.47) GRIN1GRIN2AHDAC4GRIN2BSLC6A4
SCHEMBL31426693 0.81 HDAC4 (0.47) GRIN1GRIN2AHDAC4GRIN2BSLC6A4
SCHEMBL21451950 0.81 HDAC4 (0.39) BDKRB1GRIN1GRIN2AHDAC4GRIN2B
SCHEMBL21451939 0.81 HDAC4 (0.36) BDKRB1GRIN1GRIN2AHDAC4GRIN2B
SCHEMBL21451902 0.80 HDAC4 (0.40) BDKRB1GRIN1GRIN2AHDAC4GRIN2B
SCHEMBL21452370 0.80 HDAC4 (0.47) GRIN1GRIN2AHDAC4GRIN2BPPIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed