SCHEMBL23002199

SCHEMBL23002199

Cc1ccc(F)c(C2(NC(=O)OC(C)(C)C)CCCC(O)C2=O)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 4/20 0.34
LMNA P02545 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GLA P06280 1/20 0.32
DDB1 Q16531 2/20 0.32
CRBN Q96SW2 2/20 0.32
FFAR4 Q5NUL3 1/20 0.31
DPP8 Q6V1X1 2/20 0.31
DPP9 Q86TI2 2/20 0.31
RORC P51449 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PSEN1 P49768 2/20 0.31
APP P05067 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
DRD2 P14416 1/20 0.31
ADRA2B P18089 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452558 0.90 PSEN1 (0.35) BDKRB1PSEN1APPHTR1AADRA2A
SCHEMBL21451923 0.86 FFAR4 (0.36) FFAR4TMEM97SIGMAR1BRAF
SCHEMBL21451915 0.85 BDKRB1 (0.36) BDKRB1PSEN1APPHTR1AADRA2A
SCHEMBL23002201 0.83 BDKRB1 (0.35) BDKRB1LMNAOPRK1
SCHEMBL23490927 0.83 PSEN1 (0.35) LMNANPSR1DDB1CRBNRORC
SCHEMBL21452175 0.82 HDAC4 (0.39) BDKRB1DDB1CRBNRORCCYP3A4
SCHEMBL21451948 0.82 RIPK1 (0.33) BDKRB1DDB1CRBNDPP8DPP9
SCHEMBL21452516 0.82 DDB1 (0.35) BDKRB1DDB1CRBNDPP8DPP9
SCHEMBL21451903 0.82 DDB1 (0.36) BDKRB1DDB1CRBNRORCPSEN1
SCHEMBL23490930 0.82 DDB1 (0.35) BDKRB1DDB1CRBNDPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed