SCHEMBL23011982

SCHEMBL23011982

COC(=O)c1cc2c(cc1F)C(C)(C)CC(=O)N2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.45
HDAC3 O15379 6/20 0.42
HDAC4 P56524 6/20 0.42
HDAC1 Q13547 6/20 0.42
HDAC2 Q92769 6/20 0.42
HDAC8 Q9BY41 6/20 0.42
HDAC6 Q9UBN7 6/20 0.42
HDAC9 Q9UKV0 6/20 0.42
RARB P10826 3/20 0.41
RARG P13631 3/20 0.41
TNKS O95271 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
RXRA P19793 2/20 0.34
RARA P10276 1/20 0.34
CRBN Q96SW2 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17276170 0.86 MAP3K5 (0.43) MAP3K5HDAC3HDAC4HDAC1HDAC2
SCHEMBL29706809 0.83 MAP3K5 (0.44) MAP3K5HDAC3HDAC4HDAC1HDAC2
SCHEMBL29267763 0.80 SIRT6 (0.40) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL259844 0.76 SMYD3 (0.43) HDAC3ALDH1A1LMNACRBNCCNB2
SCHEMBL23590705 0.75 RARB (0.57) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL29706811 0.75 CRBN (0.51) MAP3K5CRBNPKM
SCHEMBL3791967 0.74 RARB (0.44) MAP3K5HDAC3HDAC4HDAC1HDAC2
SCHEMBL29706774 0.74 HDAC3 (0.41) MAP3K5HDAC3HDAC4HDAC1HDAC2
SCHEMBL17276293 0.74 HDAC3 (0.41) MAP3K5HDAC3HDAC4HDAC1HDAC2
SCHEMBL23011959 0.74 MAP3K5 (0.47) MAP3K5HDAC3HDAC4HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114585616-B Amide derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-01-16 CN disclosed
CN-114585616-A Amide derivatives and their use in medicine 广东东阳光药业有限公司 2022-06-03 CN disclosed
WO-2021031071-A1 AMIDE DERIVATIVE AND USE THEREOF IN MEDICINE 广东东阳光药业有限公司 2021-02-25 WO disclosed