SCHEMBL23012008

SCHEMBL23012008

NC(=O)c1ccc2c(c1)N=CCC2

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.41
TSHR P16473 1/20 0.38
HSD17B3 P37058 1/20 0.37
LCK P06239 1/20 0.36
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
PARP1 P09874 5/20 0.34
CDC7 O00311 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
TRPA1 O75762 1/20 0.33
NNMT P40261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28039596 0.87 KDM1A (0.43) KDM1ATSHRHSD17B3LCKMKNK1
SCHEMBL27640042 0.74 ALDH1A1 (0.36) KDM4EALDH1A1TRPA1SMN1; SMN2
SCHEMBL22900627 0.73 MEN1 (0.38) KDM4EALDH1A1HSD17B10OPRM1SMN1; SMN2
SCHEMBL27730909 0.73 PBRM1 (0.37) OPRK1
SCHEMBL28413209 0.72 LCK (0.39) KDM1ATSHRHSD17B3LCKMKNK1
SCHEMBL25171204 0.71 ALDH1A1 (0.49) KDM1ATSHRKDM4EALDH1A1HSD17B10
SCHEMBL29790728 0.71 KMT2A (0.36) TSHRLCKMKNK1MKNK2KDM4E
SCHEMBL21168435 0.70 HSD17B3 (0.55) KDM1ATSHRHSD17B3LCKKDM4E
SCHEMBL19691161 0.70 CDC7 (0.41) TSHRLCKMKNK1MKNK2SIRT2
SCHEMBL4433792 0.70 TSHR (0.53) TSHRLCKMKNK1MKNK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021031071-A1 AMIDE DERIVATIVE AND USE THEREOF IN MEDICINE 广东东阳光药业有限公司 2021-02-25 WO disclosed