SCHEMBL23017405

SCHEMBL23017405

NC(=O)c1c[nH]c(CO)c(OCc2ccccc2)c1=O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.46
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
MDH2 P40926 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PARP1 P09874 1/20 0.43
SIRT2 Q8IXJ6 2/20 0.41
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GSTP1 P09211 1/20 0.37
LMNA P02545 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16587496 0.87 SMN1; SMN2 (0.46) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL12993083 0.85 ALDH1A1 (0.49) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL16437764 0.80 POLB (0.49) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL19853588 0.75 ALDH1A1 (0.49) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL18473801 0.74 KCNA5 (0.52) ALDH1A1HPGDSMN1; SMN2POLBHTT
SCHEMBL18567041 0.71 SMN1; SMN2 (0.48) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL19730907 0.71 SIRT2 (0.50) PARP10ALDH1A1HPGDSMN1; SMN2PARP1
SCHEMBL5264504 0.70 MAPK14 (0.45) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL16587510 0.70 ALDH1A1 (0.47) ALDH1A1HPGDMDH2SMN1; SMN2POLB
SCHEMBL19706906 0.69 MAPK14 (0.46) ALDH1A1HPGDMDH2SMN1; SMN2GSTP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3456721-B1 METHOD OF PRODUCING COMPOUNDS HAVING HIV INTEGRASE INHIVITORY ACTIVITY SHIONOGI & CO (JP) 2021-02-24 EP disclosed