SCHEMBL2301871

SCHEMBL2301871

C=CC(=O)N1CCN(Cc2ccc(CCOc3ccc(C(C)C)cc3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.54
ALDH1A1 P00352 2/20 0.54
HTT P42858 1/20 0.54
HRH3 Q9Y5N1 1/20 0.53
GPR183 P32249 1/20 0.53
FAAH O00519 3/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
POLB P06746 1/20 0.46
PKM P14618 1/20 0.46
PPARG P37231 1/20 0.45
PPARD Q03181 1/20 0.45
PPARA Q07869 1/20 0.45
IDH1 O75874 3/20 0.45
IDH2 P48735 3/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2297065 0.99 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1HTTHRH3GPR183
SCHEMBL14108437 0.89 DRD3 (0.49) SMN1; SMN2ALDH1A1HRH3GPR183FAAH
SCHEMBL2231731 0.88 HRH3 (0.58) SMN1; SMN2ALDH1A1HTTHRH3GPR183
SCHEMBL2232804 0.88 HRH3 (0.58) SMN1; SMN2ALDH1A1HTTHRH3GPR183
SCHEMBL22185391 0.87 ALDH1A1 (0.68) SMN1; SMN2ALDH1A1HTTHRH3GPR183
SCHEMBL13582370 0.84 HRH3 (0.60) SMN1; SMN2ALDH1A1HTTHRH3FAAH
SCHEMBL2233177 0.82 HRH3 (0.57) SMN1; SMN2ALDH1A1HTTHRH3GPR183
SCHEMBL14110188 0.82 HRH3 (0.51) SMN1; SMN2ALDH1A1HTTHRH3FAAH
SCHEMBL14108479 0.82 KDM4E (0.61) SMN1; SMN2ALDH1A1HRH3FAAHMEN1
SCHEMBL2234825 0.78 HRH3 (0.51) HRH3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528897-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS Otsuka Pharmaceutical Co., Ltd. (JP) 2012-12-05 EP claimed
WO-2011093524-A9 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-12-01 WO claimed
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO claimed