SCHEMBL2302769

SCHEMBL2302769

COc1ccccc1-c1nc[nH]n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
HSD17B10 Q99714 3/20 0.50
GAA P10253 1/20 0.50
DCUN1D1 Q96GG9 2/20 0.49
METAP2 P50579 1/20 0.49
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2D6 P10635 3/20 0.47
ALPL P05186 1/20 0.47
XDH P47989 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 2/20 0.45
TP53 P04637 2/20 0.45
RAB9A P51151 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 1/20 0.45
MAPK1 P28482 1/20 0.45
PPARG P37231 1/20 0.45
KMT2A Q03164 1/20 0.45
NCOA2 Q15596 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288342 0.84 LRRK2 (0.44) HSD17B10CYP1A2CYP3A4CYP2D6SMN1; SMN2
SCHEMBL15125436 0.77 GAA (0.52) ALDH1A1HSD17B10GAADCUN1D1METAP2
SCHEMBL10801976 0.77 DCUN1D1 (0.43) ALDH1A1DCUN1D1SMN1; SMN2NPC1RAB9A
SCHEMBL16790012 0.76 CYP1A2 (0.62) ALDH1A1HSD17B10GAACYP1A2CYP3A4
SCHEMBL12127343 0.76 ALDH1A1 (0.50) ALDH1A1HSD17B10SMN1; SMN2NPC1RAB9A
SCHEMBL23066466 0.76 ALDH1A1 (0.61) ALDH1A1HSD17B10GAADCUN1D1CYP1A2
SCHEMBL17194909 0.75 BRD4 (0.36) ALDH1A1HSD17B10GAADCUN1D1CYP1A2
SCHEMBL2099637 0.75 IDO1 (0.48) ALDH1A1CYP1A2CYP3A4CYP2D6SMN1; SMN2
SCHEMBL9173243 0.73 IDO1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2D6SMN1; SMN2
SCHEMBL174453 0.73 CYP1A2 (0.54) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103016-A2 COMPOSITIONS AND METHODS FOR INHIBITING EZH2 THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2011-08-25 WO disclosed