SCHEMBL2303041

SCHEMBL2303041

Cc1ccc(NC(=O)c2ccc(N3CCN(C(=O)NCCC(=O)O)CC3)nc2)cc1I

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 1/20 0.47
RAB9A P51151 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
KLK7 P49862 1/20 0.42
MAPT P10636 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
FOLH1 Q04609 1/20 0.42
TRPV1 Q8NER1 2/20 0.42
HDAC1 Q13547 2/20 0.41
PANK3 Q9H999 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
FASN P49327 1/20 0.41
POLB P06746 1/20 0.40
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301002 0.90 P2RY12 (0.50) P2RY12RAB9AL3MBTL1KMT2AMAPT
SCHEMBL3310147 0.89 P2RY12 (0.49) P2RY12RAB9AL3MBTL1KMT2AMEN1
SCHEMBL3308028 0.84 P2RY12 (0.51) P2RY12RAB9AL3MBTL1KMT2AMAPT
SCHEMBL2357597 0.84 KDM4E (0.49) P2RY12RAB9AL3MBTL1MAPTCYP1A2
SCHEMBL3311413 0.83 USP30 (0.53) P2RY12RAB9AL3MBTL1KMT2AMAPT
SCHEMBL13363955 0.82 KCNQ3 (0.57) RAB9AL3MBTL1MAPTCYP1A2CYP2C19
SCHEMBL2305153 0.82 RAB9A (0.49) RAB9AL3MBTL1MAPTCYP1A2CYP2C19
SCHEMBL2300887 0.81 RAB9A (0.47) P2RY12RAB9AL3MBTL1MAPTCYP1A2
SCHEMBL2357220 0.81 RAB9A (0.45) P2RY12RAB9AL3MBTL1KMT2AMEN1
SCHEMBL2356882 0.81 RAB9A (0.50) RAB9AL3MBTL1KMT2AMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350311-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS Via Pharmaceuticals, Inc. (US) 2011-08-03 EP disclosed
WO-2010056506-A1 DIACYLGLYCEROL ACLYTRANSFERASE INHIBITORS VIA PHARMACEUTICALS, INC. (US) 2010-05-20 WO disclosed