SCHEMBL2303446

SCHEMBL2303446

O=C1CCC(c2cccc(Cl)c2)C(=O)O1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.43
TP53 P04637 3/20 0.42
MAPT P10636 2/20 0.42
MDM2 Q00987 4/20 0.42
LMNA P02545 1/20 0.41
SLC6A3 Q01959 4/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
SLC6A2 P23975 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11329173 0.89 CTRB1 (0.49) CTRB1TP53MAPTLMNANPSR1
SCHEMBL6781180 0.81 CYP19A1 (0.46) CTRB1SLC6A3ALDH1A1SLC6A2
SCHEMBL26448018 0.81 SIRT2 (0.46) CTRB1MAPTLMNANPSR1ALDH1A1
SCHEMBL9541605 0.80 CTRB1 (0.44) CTRB1TP53MAPTLMNASLC6A3
SCHEMBL192372 0.80 CTRB1 (0.63) CTRB1TP53MAPTLMNAGAA
SCHEMBL7815009 0.79 SLC6A2 (0.41) CTRB1TP53MAPTLMNASLC6A3
SCHEMBL9435442 0.77 CTRB1 (0.50) CTRB1TP53MAPTLMNANPSR1
SCHEMBL28730826 0.74 MDM2 (0.43) TP53MAPTMDM2SLC6A3ALDH1A1
SCHEMBL28730828 0.74 MDM2 (0.43) TP53MAPTMDM2SLC6A3ALDH1A1
SCHEMBL29576656 0.74 MDM2 (0.43) TP53MAPTMDM2SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349999-A1 ALLOSTERIC PROTEIN KINASE MODULATORS Universität des Saarlandes (DE) 2011-08-03 EP disclosed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed
WO-1998002432-A1 BICYCLIC COMPOUNDS FOR CONTROLLING MICTURITION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-22 WO disclosed