SCHEMBL23049685

SCHEMBL23049685

COCCOC(=O)C(C)(C)N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
ALDH1A1 P00352 3/20 0.36
GAA P10253 3/20 0.36
RAB9A P51151 1/20 0.36
POLB P06746 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
RECQL P46063 1/20 0.35
XIAP P98170 1/20 0.35
KMT2A Q03164 1/20 0.35
PLEC Q15149 1/20 0.35
ADORA2A P29274 1/20 0.35
FDPS P14324 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ARG1 P05089 1/20 0.33
ARG2 P78540 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15679087 0.91 POLB (0.33) TSHRALDH1A1GAAPOLBNPSR1
SCHEMBL4156487 0.81 POLB (0.43) TSHRALDH1A1GAAPOLBNPSR1
SCHEMBL31629763 0.79 TSHR (0.41) TSHRALDH1A1GAARAB9APOLB
SCHEMBL2302371 0.79 HCAR2 (0.39) TSHRALDH1A1RAB9AMEN1MAPT
SCHEMBL15658014 0.79 TSHR (0.38) TSHRALDH1A1GAAPOLBNPSR1
SCHEMBL18274690 0.79 ALDH1A1 (0.35) ALDH1A1GAAPOLBNPSR1MAPT
SCHEMBL21305791 0.78 ALDH1A1 (0.54) TSHRALDH1A1POLBMAPTTHRB
SCHEMBL4608266 0.77 TSHR (0.44) TSHRALDH1A1GAARAB9APOLB
SCHEMBL18842478 0.77 TSHR (0.39) TSHRALDH1A1GAAPOLBNPSR1
SCHEMBL14280608 0.77 TSHR (0.39) TSHRALDH1A1GAAPOLBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3596064-B1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-03-03 EP disclosed