SCHEMBL2305446

SCHEMBL2305446

CSC(=S)Oc1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTH P32929 1/20 0.40
KDM4E B2RXH2 4/20 0.37
LMNA P02545 3/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
METAP1 P53582 1/20 0.37
BLM P54132 1/20 0.37
HIF1A Q16665 1/20 0.37
DOHH Q9BU89 1/20 0.37
P4HTM Q9NXG6 1/20 0.37
NPC1 O15118 6/20 0.36
RAB9A P51151 6/20 0.36
SMN1; SMN2 Q16637 5/20 0.36
ALDH1A1 P00352 3/20 0.36
TP53 P04637 2/20 0.36
HPGD P15428 2/20 0.36
HTT P42858 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3872197 0.79 EHMT2 (0.44) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL19435589 0.79 KDM4E (0.41) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL435144 0.78 KDM4E (0.44) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL31734268 0.78 KDM4E (0.44) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL670301 0.76 KDM4E (0.42) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL11121873 0.75 NOS3 (0.43) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL10416676 0.75 NOS3 (0.43) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL27936240 0.75 KDM4E (0.41) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL6502675 0.75 KDM4E (0.41) KDM4ELMNACYP1A2POLBCCR1
SCHEMBL5577241 0.75 KDM4E (0.41) KDM4ELMNACYP1A2POLBCCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350008-B1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES BAYER CROPSCIENCE AG (DE) 2012-09-05 EP disclosed
EP-2350008-A1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES Bayer CropScience AG (DE) 2011-08-03 EP disclosed
WO-2010040461-A1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES BAYER CROPSCIENCE AG (DE) 2010-04-15 WO disclosed