SCHEMBL2306574

SCHEMBL2306574

O=C(O)C(Cc1c[nH]c2ccc(F)cc12)Nc1ccc2cc(Cl)ccc2n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 4/20 0.46
ICAM1 P05362 4/20 0.46
ITGAL P20701 4/20 0.46
TSHR P16473 1/20 0.44
ADAM17 P78536 1/20 0.43
CCKBR P32239 1/20 0.43
SNCA P37840 3/20 0.42
HTR2A P28223 2/20 0.41
HTR2C P28335 1/20 0.41
PPARG P37231 1/20 0.41
NOTUM Q6P988 2/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
MPO P05164 2/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2309016 0.93 ITGB2 (0.46) ITGB2ICAM1ITGALADAM17PPARG
SCHEMBL2309696 0.89 ITGB2 (0.44) ITGB2ICAM1ITGALTSHRADAM17
SCHEMBL2312170 0.85 ITGB2 (0.47) ITGB2ICAM1ITGALTSHRADAM17
SCHEMBL2311993 0.78 ITGB2 (0.47) ITGB2ICAM1ITGALADAM17PPARG
SCHEMBL2306893 0.77 ITGB2 (0.54) ITGB2ICAM1ITGALPPARG
SCHEMBL28163340 0.75 TSHR (0.60) ITGB2ICAM1ITGALTSHRADAM17
SCHEMBL30138755 0.74 TSHR (0.59) ITGB2ICAM1ITGALTSHRADAM17
SCHEMBL5056897 0.74 TSHR (0.59) ITGB2ICAM1ITGALTSHRADAM17
SCHEMBL2310201 0.74 ITGB2 (0.44) ITGB2ICAM1ITGALADAM17HTR2A
SCHEMBL2313903 0.73 NHERF1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350014-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2011-08-03 EP claimed
EP-2350014-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2011-08-03 EP disclosed