SCHEMBL23073664

SCHEMBL23073664

Nc1ccnc(-c2cnc(N3CCCCC3)nc2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 3/20 0.41
CDC42BPB Q9Y5S2 3/20 0.41
ROCK2 O75116 2/20 0.41
PIK3R1 P27986 3/20 0.40
PIK3CA P42336 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MTOR P42345 2/20 0.40
CNR2 P34972 3/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CB P42338 1/20 0.39
DHFR P00374 1/20 0.38
CDC42BPA Q5VT25 1/20 0.37
DYRK1A Q13627 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17210409 0.98 PIK3CA (0.40) ROCK1CDC42BPBROCK2PIK3R1PIK3CA
SCHEMBL17202011 0.83 GSK3A (0.37) ROCK2PIK3R1PIK3CAMTORPIK3CD
SCHEMBL17202046 0.79 DYRK1A (0.41) PIK3R1PIK3CAMTORDYRK1A
SCHEMBL18539061 0.79 MTOR (0.38) PIK3R1PIK3CAALDH1A1MTORDYRK1A
SCHEMBL17201976 0.79 MAP3K12 (0.34) ROCK2PIK3R1PIK3CAMTORPIK3CD
SCHEMBL17210337 0.79 CNR2 (0.45) ALDH1A1CNR2NPC1RAB9AKDM4E
SCHEMBL9900073 0.79 KDM1A (0.47) ROCK1CDC42BPBROCK2PIK3R1PIK3CA
SCHEMBL21861329 0.77 MTOR (0.36) PIK3R1PIK3CAMTOR
SCHEMBL17210359 0.77 MAP3K12 (0.43) ALDH1A1DYRK1AKDM4EHPGDALOX15
SCHEMBL17210367 0.77 KDM4E (0.43) ALDH1A1CNR2DYRK1AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3134410-B1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL LILLY CO ELI (US) 2021-03-10 EP disclosed