SCHEMBL2308124

SCHEMBL2308124

CCC(CC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)OCCOC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP3A4 P08684 3/20 0.40
MAOA P21397 2/20 0.40
TSHR P16473 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PDE4D Q08499 1/20 0.40
RAB9A P51151 2/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2D6 P10635 2/20 0.37
HTR3A P46098 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
BLM P54132 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PHLPP2 Q6ZVD8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1747948 0.84 KMT2A (0.51) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL1748271 0.76 NPC1 (0.55) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL5068457 0.76 KMT2A (0.52) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL1747972 0.76 KMT2A (0.52) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL6031378 0.73 NPC1 (0.58) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL1748086 0.73 NPC1 (0.58) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL5068844 0.72 NPC1 (0.60) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL4226578 0.72 NPC1 (0.60) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL4229648 0.72 LMNA (0.54) NPC1KMT2AMEN1LMNACYP1A2
SCHEMBL5068496 0.72 KMT2A (0.57) NPC1KMT2AMEN1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP disclosed