SCHEMBL2309348

SCHEMBL2309348

COC(c1ccc(F)cc1)C1(C(C(=O)Nc2ccc(C(=O)O)cn2)C2CCCCC2)Nc2cc(F)c(F)cc2N1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GCK P35557 11/20 0.45
NR1H4 Q96RI1 2/20 0.44
HCAR3 P49019 3/20 0.39
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC2 Q92769 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2308317 0.94 NR1H4 (0.45) GCKNR1H4HCAR3HDAC3HDAC2
SCHEMBL2305479 0.94 NR1H4 (0.45) GCKNR1H4HCAR3HDAC3HDAC2
SCHEMBL2308785 0.88 NR1H4 (0.40) NR1H4
SCHEMBL2308591 0.87 NR1H4 (0.43) NR1H4
SCHEMBL2305595 0.85 NR1H4 (0.49) NR1H4KMT2A
SCHEMBL2310551 0.85 NR1H4 (0.41) NR1H4MEN1KMT2A
SCHEMBL2304490 0.83 NR1H4 (0.44) NR1H4
SCHEMBL2309699 0.83 NR1H4 (0.39) NR1H4
SCHEMBL2306822 0.82 NR1H4 (0.41) NR1H4MEN1KMT2A
SCHEMBL2307306 0.82 NR1H4 (0.41) NR1H4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350022-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-08-03 EP claimed
WO-2010043513-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-04-22 WO claimed
EP-2350022-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-08-03 EP disclosed
WO-2010043513-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-04-22 WO disclosed