SCHEMBL23097565

SCHEMBL23097565

O=C1Cc2cc(OCCCN3CCN(c4ccc(-c5ccccc5)cc4)CC3)ccc2N1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.63
DRD3 P35462 7/20 0.58
HTR1A P08908 4/20 0.58
HTR2A P28223 4/20 0.58
SLC6A4 P31645 3/20 0.58
DRD4 P21917 2/20 0.58
HTR2C P28335 2/20 0.58
HTR7 P34969 2/20 0.58
KCNH2 Q12809 1/20 0.55
MAOA P21397 2/20 0.53
MAOB P27338 2/20 0.53
HRH1 P35367 2/20 0.53
TMEM97 Q5BJF2 2/20 0.53
SIGMAR1 Q99720 2/20 0.53
KDM1A O60341 1/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
HRH3 Q9Y5N1 1/20 0.52
SLC6A2 P23975 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10489982 0.95 DRD2 (0.69) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097631 0.92 DRD2 (0.72) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097667 0.89 DRD3 (0.60) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097697 0.88 KCNH2 (0.58) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097637 0.88 DRD2 (0.58) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097632 0.88 MAOB (0.64) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097771 0.88 SLC6A4 (0.61) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097620 0.88 KCNH2 (0.69) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097761 0.88 DRD2 (0.65) DRD2DRD3HTR1AHTR2ASLC6A4
SCHEMBL23097614 0.87 DRD2 (0.59) DRD2DRD3HTR1AHTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170334-B1 NMDA RECEPTOR ANTAGONISTS FOR NEUROPROTECTION UNIV EMORY (US) 2021-03-17 EP disclosed