SCHEMBL2310643

SCHEMBL2310643

Cc1ccc(Nc2ccccn2)cc1-c1ccc(NC(=O)c2c(F)cccc2F)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL2 P60568 15/20 0.57
JAK2 O60674 2/20 0.46
JAK1 P23458 2/20 0.46
TYK2 P29597 2/20 0.46
HTT P42858 1/20 0.46
NOD2 Q9HC29 1/20 0.46
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
APEX1 P27695 1/20 0.45
TNF P01375 1/20 0.45
STIM1 Q13586 1/20 0.45
ORAI1 Q96D31 1/20 0.45
DYRK3 O43781 1/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
ABL1 P00519 1/20 0.44
EGFR P00533 1/20 0.44
NTRK1 P04629 1/20 0.44
PRKCG P05129 1/20 0.44
LCK P06239 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4764906 0.85 IL2 (0.60) IL2JAK2JAK1TYK2HTT
SCHEMBL2313336 0.80 IL2 (0.54) IL2JAK2JAK1TYK2HTT
SCHEMBL1828207 0.80 IL2 (0.63) IL2JAK2JAK1TYK2HTT
SCHEMBL2311041 0.79 IL2 (0.53) IL2
SCHEMBL4766353 0.79 IL2 (0.63) IL2JAK2JAK1TYK2HTT
SCHEMBL4770059 0.79 IL2 (0.62) IL2JAK2JAK1TYK2HTT
SCHEMBL12093752 0.78 IL2 (0.57) IL2JAK2JAK1TYK2HTT
SCHEMBL4762567 0.77 IL2 (0.71) IL2JAK2JAK1TYK2HTT
SCHEMBL4764710 0.77 IL2 (0.58) IL2JAK2JAK1TYK2HTT
SCHEMBL16471113 0.77 IL2 (0.63) IL2JAK2JAK1TYK2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120196838-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2012-08-02 US claimed
US-20100130522-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-05-27 US claimed
US-20140045861-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2014-02-13 US disclosed
US-20140045861-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2014-02-13 US disclosed
US-20120196838-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2012-08-02 US disclosed
US-20120196838-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2012-08-02 US disclosed
EP-2350006-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES Synta Pharmaceuticals Corp. (US) 2011-08-03 EP disclosed
US-20100130522-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-05-27 US disclosed
US-20100130522-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-05-27 US disclosed
US-20100130522-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-05-27 US disclosed
WO-2010039238-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-04-08 WO disclosed
WO-2010039238-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-04-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120196838-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES CCR1, CXCL8, CCR9 IL2 7/4885JAK2 1811/4885JAK1 1223/4885
US-20100130522-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES CCR1, CXCL8, CCR9 IL2 7/4885JAK2 1811/4885JAK1 1223/4885
US-20140045861-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES CCR1, CXCL8, CCR9 IL2 7/4885JAK2 1811/4885JAK1 1223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.