Bicarbonate

Bicarbonate

SCHEMBL2311617

O=C(O)O.O=C(c1ccc(-c2ccc(Nc3nc4cc(F)ccc4s3)cc2)cc1)C1CCCC1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.51
CSGALNACT1 Q8TDX6 1/20 0.50
DYRK1A Q13627 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
MAPT P10636 2/20 0.44
CSF1R P07333 2/20 0.44
HCRTR1 O43613 2/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
TNF P01375 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
NR2F2 P24468 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
KLF5 Q13887 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL2307791 0.92 DGAT1 (0.61) DGAT1CSGALNACT1DYRK1ASMN1; SMN2NPC1
Bicarbonate SCHEMBL2314526 0.89 DGAT1 (0.67) DGAT1CSGALNACT1DYRK1ASMN1; SMN2NPC1
Bicarbonate SCHEMBL2307044 0.88 CSF1R (0.44) DGAT1CSGALNACT1MAPTCSF1RHCRTR1
Bicarbonate SCHEMBL2309849 0.87 DYRK1A (0.48) DGAT1CSGALNACT1DYRK1AMAPTCSF1R
SCHEMBL1748021 0.86 DGAT1 (0.69) DGAT1CSGALNACT1DYRK1AHCRTR1
SCHEMBL1748022 0.86 DGAT1 (0.69) DGAT1CSGALNACT1DYRK1AHCRTR1
SCHEMBL1748020 0.86 DGAT1 (0.69) DGAT1CSGALNACT1DYRK1AHCRTR1
SCHEMBL12266127 0.86 DGAT1 (0.69) DGAT1CSGALNACT1DYRK1AHCRTR1
Bicarbonate SCHEMBL2311438 0.86 DGAT1 (0.45) DGAT1CSGALNACT1SMN1; SMN2RAB9AMAPT
Bicarbonate SCHEMBL2310107 0.85 NPC1 (0.53) SMN1; SMN2NPC1RAB9AMAPTCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP claimed