SCHEMBL23127

SCHEMBL23127

COc1cccc(C(=O)c2cc(Br)cs2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
PARP1 P09874 1/20 0.51
STS P08842 2/20 0.50
MAPK13 O15264 1/20 0.48
MAPK12 P53778 1/20 0.48
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
POLB P06746 1/20 0.47
CASP3 P42574 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
HPGD P15428 1/20 0.46
CNR2 P34972 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534530 0.81 CES2 (0.52) CES2CES1PARP1POLBNPC1
SCHEMBL4238012 0.80 CES2 (0.62) CES2CES1PARP1STSNPC1
SCHEMBL30136061 0.80 CES2 (0.62) CES2CES1PARP1STSNPC1
SCHEMBL22718 0.79 POLB (0.67) CES2CES1PARP1STSMAPK13
SCHEMBL23041066 0.79 NPC1 (0.65) CES2CES1PARP1STSNPC1
SCHEMBL31414638 0.79 CES2 (0.77) CES2CES1PARP1STSNPC1
SCHEMBL4823687 0.79 CES2 (0.77) CES2CES1PARP1STSNPC1
SCHEMBL18529835 0.78 CES2 (0.61) CES2CES1PARP1STSNPC1
SCHEMBL3468157 0.78 KMT2A (0.69) CES2CES1PARP1STSNPC1
SCHEMBL31291512 0.78 KMT2A (0.69) CES2CES1PARP1STSNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed