SCHEMBL23158698

SCHEMBL23158698

O=c1c(CO)c[nH]cc1-c1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.38
CDK4 P11802 2/20 0.37
CCND1 P24385 2/20 0.37
ERCC1 P07992 2/20 0.37
ERCC4 Q92889 2/20 0.37
GRM2 Q14416 2/20 0.36
BCL2L1 Q07817 1/20 0.36
BAD Q92934 1/20 0.36
PTGS1 P23219 1/20 0.35
SERPINE1 P05121 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
PPARG P37231 1/20 0.34
RAB9A P51151 1/20 0.34
PPARD Q03181 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14949020 0.86 MAPT (0.36) NR4A2ERCC1ERCC4SLC6A4SLC6A3
SCHEMBL28199937 0.85 NR4A2 (0.33) NR4A2CDK4CCND1ERCC1ERCC4
SCHEMBL363193 0.79 KDM4E (0.46) BCL2L1BADSLC6A4SLC6A3KDM4E
SCHEMBL28319846 0.77 SLC6A4 (0.38) NR4A2BCL2L1BADPTGS1SLC6A4
SCHEMBL20351754 0.75 BRD4 (0.40) NR4A2ERCC1ERCC4BCL2L1BAD
SCHEMBL18031340 0.75 NR4A2 (0.40) NR4A2ERCC1ERCC4GRM2BCL2L1
SCHEMBL28199967 0.75 GRM2 (0.36) NR4A2ERCC1ERCC4GRM2BCL2L1
SCHEMBL17233734 0.75 AURKB (0.42) ERCC1ERCC4BCL2L1BADPTGS1
SCHEMBL29757272 0.75 IKBKB (0.43) GRM2PTGS1SLC6A4SLC6A3AURKB
SCHEMBL10396846 0.74 NR4A2 (0.47) NR4A2ERCC1ERCC4BCL2L1BAD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3168219-B1 PYRIDONE DERIVATIVE HAVING TETRAHYDROPYRANYL METHYL GROUP DAIICHI SANKYO CO LTD (JP) 2021-03-31 EP disclosed