SCHEMBL2316320

SCHEMBL2316320

CC(=O)C=CC1=CC(C)(C)COc2cc(Br)c(F)cc21

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.34
MAOB P27338 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2316311 1.00 AKR1B1 (0.34) AKR1B1MAOBESR1ESR2
SCHEMBL2317446 0.86 NOTUM (0.37) AKR1B1ESR1ESR2
SCHEMBL2317447 0.86 NOTUM (0.37) AKR1B1ESR1ESR2
SCHEMBL2317337 0.82 MEN1 (0.31)
SCHEMBL2317332 0.82 MEN1 (0.31)
SCHEMBL2314394 0.81 APP (0.34) MAOB
SCHEMBL2314398 0.81 APP (0.34) MAOB
SCHEMBL2316995 0.81 ALDH1A1 (0.39) AKR1B1MAOBESR1ESR2
SCHEMBL2316992 0.81 ALDH1A1 (0.39) AKR1B1MAOBESR1ESR2
SCHEMBL2315821 0.79 KDM4E (0.39) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP claimed