SCHEMBL2316677

SCHEMBL2316677

CC(C)OC(=O)N(c1ccc(F)c(-c2nn(CCF)cc2-c2ccncc2)c1F)S(=O)(=O)c1cc(F)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.35
SLC6A3 Q01959 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2359853 0.93 BRAF (0.33)
SCHEMBL2316981 0.92 SLC6A3 (0.37) PDE10ASLC6A3
SCHEMBL2359701 0.90 PDE10A (0.37) PDE10ASLC6A3
SCHEMBL2359382 0.90 PSEN1 (0.35)
SCHEMBL2359183 0.90 CSNK1D (0.40) PDE10A
SCHEMBL2319490 0.89 PDE10A (0.36) PDE10ASLC6A3
SCHEMBL2318287 0.89 PDE10A (0.34) PDE10ASLC6A3
SCHEMBL14719049 0.87 PDE10A (0.34) PDE10ASLC6A3
SCHEMBL2358909 0.86 BRAF (0.38)
SCHEMBL2359191 0.84 BRAF (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528909-A1 SULFONAMIDO DERIVATIVES OF 3,4-DIARYLPYRAZOLES AS PROTEIN KINASE INHIBITORS Nerviano Medical Sciences S.r.l. (IT) 2012-12-05 EP claimed
WO-2011092088-A1 SULFONAMIDO DERIVATIVES OF 3,4-DIARYLPYRAZOLES AS PROTEIN KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2011-08-04 WO claimed
EP-2528909-B1 SULFONAMIDO DERIVATIVES OF 3,4-DIARYLPYRAZOLES AS PROTEIN KINASE INHIBITORS NERVIANO MEDICAL SCIENCES SRL (IT) 2016-06-22 EP disclosed
WO-2011092088-A1 SULFONAMIDO DERIVATIVES OF 3,4-DIARYLPYRAZOLES AS PROTEIN KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2011-08-04 WO disclosed