SCHEMBL2316808

SCHEMBL2316808

Clc1cc(Cl)c2nc[nH]c2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.34
PIM1 P11309 3/20 0.34
AURKA O14965 2/20 0.34
DAPK3 O43293 2/20 0.34
PRKD3 O94806 2/20 0.34
MAP4K4 O95819 2/20 0.34
RET P07949 2/20 0.34
IGF1R P08069 2/20 0.34
CLK2 P49760 2/20 0.34
GSK3A P49840 2/20 0.34
GSK3B P49841 2/20 0.34
PRKX P51817 2/20 0.34
BTK Q06187 2/20 0.34
TYRO3 Q06418 2/20 0.34
DYRK1A Q13627 2/20 0.34
NTRK3 Q16288 2/20 0.34
TAOK1 Q7L7X3 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
ALK Q9UM73 2/20 0.34
JAK2 O60674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29574753 1.00 CSNK2A1 (0.34) CSNK2A1PIM1AURKADAPK3PRKD3
SCHEMBL16774129 0.80 CSNK2A1 (0.40) CSNK2A1PIM1AURKADAPK3PRKD3
SCHEMBL26106496 0.80 PARP1 (0.40) CSNK2A1PIM1PARP1PIM2AXL
SCHEMBL31347215 0.80 MEN1 (0.36) CSNK2A1PIM1IGF1RCLK2GSK3A
SCHEMBL30611884 0.80 PARP1 (0.40) CSNK2A1PIM1PARP1PIM2AXL
SCHEMBL10399191 0.80 DPP4 (0.34) CSNK2A1PIM1AURKADAPK3PRKD3
SCHEMBL22757469 0.80 PIM1 (0.36) CSNK2A1PIM1AURKADAPK3PRKD3
SCHEMBL10626643 0.71 CDK2 (0.39) AURKAGSK3BABL1METCDK7
SCHEMBL18114683 0.69 MAPT (0.42) LRRK2MAPTKDM4EGAA
SCHEMBL127024 0.68 AXL (0.48) CSNK2A1PIM1AURKADAPK3PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 107 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125378-A2 Heterocyclic Compounds BEONE MEDICINES I GMBH (CH) 2026-05-07 US disclosed
US-20250353846-A1 Heterocyclic Compounds BEONE MEDICINES I GMBH (CH) 2025-11-20 US disclosed
EP-4634186-A1 2,6,9-TRISUBSTITUTED PURINES Astrazeneca AB (SE) 2025-10-22 EP disclosed
US-12441744-B2 2,6,9-trisubstituted purines ASTRAZENECA AB 2025-10-14 US disclosed
US-12435095-B2 Substituted morpholines as ATR kinase inhibitors SHANGHAI ANNOVA BIOTECHNOLOGY CO., LTD. (CN) 2025-10-07 US disclosed
US-12421273-B2 Ectonucleotidase inhibitors and methods of use thereof ANTENGENE THERAPEUTICS LIMITED (CN) 2025-09-23 US disclosed
US-20250197425-A1 2,6,9-TRISUBSTITUTED PURINES ASTRAZENECA AB (SE) 2025-06-19 US disclosed
US-20250179070-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE AS ATR KINASE INHIBITORS REPARE THERAPEUTICS INC (CA) 2025-06-05 US disclosed
WO-2025080788-A1 CCR4 INHIBITORS AND METHODS OF USE THEREOF RAYTHERA, INC. (US) 2025-04-17 WO disclosed
US-12264155-B2 Compounds, pharmaceutical compositions, and methods of preparing compounds and of their use as ATR kinase inhibitors REPARE THERAPEUTICS INC. (CA) 2025-04-01 US disclosed
US-20140114070-A1 COMPOUNDS THAT EXPAND HEMATOPOIETIC STEM CELLS THE SCRIPPS RESEARCH INSTITUTE (US) 2014-04-24 US disclosed
WO-2013095761-A1 IMIDAZOPYRIDINE DERIVATIVES AS PI3 KINASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-06-27 WO disclosed
WO-2013095761-A1 IMIDAZOPYRIDINE DERIVATIVES AS PI3 KINASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-06-27 WO disclosed
EP-2350078-A2 COMPOUNDS THAT EXPAND HEMATOPOIETIC STEM CELLS IRM LLC (BM) 2011-08-03 EP disclosed
US-20100183564-A1 COMPOUNDS THAT EXPAND HEMATOPOIETIC STEM CELLS IRM LLC (BM) 2010-07-22 US disclosed
WO-2010059401-A2 COMPOUNDS THAT EXPAND HEMATOPOIETIC STEM CELLS IRM LLC (BM) 2010-05-27 WO disclosed
US-7358235-B2 Analogs of nitrobenzylthioinosine GRUENENTHAL GMBH (DE) 2008-04-15 US disclosed
US-7358235-B2 Analogs of nitrobenzylthioinosine GRUENENTHAL GMBH (DE) 2008-04-15 US disclosed
US-4780452-A ANTIINFLAMMATORY AGENTS, ANTIPYRETICS BURROUGHS WELLCOME CO. (US) 1988-10-25 US disclosed
EP-0260852-A2 Nucleoside Analogues THE WELLCOME FOUNDATION LIMITED (GB) 1988-03-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12435095-B2 Substituted morpholines as ATR kinase inhibitors ATR, WEE1, WEE2 CSNK2A1 322/4885PIM1 585/4885AURKA 64/4885
US-20260125378-A2 Heterocyclic Compounds NFATC1, CD4, MALT1 CSNK2A1 954/4885PIM1 4476/4885AURKA 2743/4885
US-12421273-B2 Ectonucleotidase inhibitors and methods of use thereof NT5E, ENTPD5, NT5C2 CSNK2A1 3460/4885PIM1 4578/4885AURKA 3513/4885
US-20250179070-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE AS ATR KINASE INHIBITORS ATR, CHEK2, CHEK1 CSNK2A1 131/4885PIM1 2762/4885AURKA 177/4885
US-20250353846-A1 Heterocyclic Compounds NFATC1, CD4, ACIN1 CSNK2A1 580/4885PIM1 1203/4885AURKA 937/4885
US-12441744-B2 2,6,9-trisubstituted purines CDK2, CDK1, CCNT2 CSNK2A1 113/4885PIM1 860/4885AURKA 147/4885
US-20250197425-A1 2,6,9-TRISUBSTITUTED PURINES CDK2, CDK1, CCNT2 CSNK2A1 113/4885PIM1 860/4885AURKA 147/4885
US-20140114070-A1 COMPOUNDS THAT EXPAND HEMATOPOIETIC STEM CELLS CD47, HCLS1, CD74 CSNK2A1 4693/4885PIM1 1708/4885AURKA 2901/4885
US-20100183564-A1 COMPOUNDS THAT EXPAND HEMATOPOIETIC STEM CELLS CD47, HCLS1, CD74 CSNK2A1 4693/4885PIM1 1708/4885AURKA 2901/4885
US-12264155-B2 Compounds, pharmaceutical compositions, and methods of preparing compounds and of their use as ATR kinase inhibitors ATR, CHEK2, CHEK1 CSNK2A1 131/4885PIM1 2762/4885AURKA 177/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.