SCHEMBL23181529

SCHEMBL23181529

Cc1ncc(C2CC2)cc1I

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
PDGFRB P09619 1/20 0.37
PDGFRA P16234 1/20 0.37
PSMB5 P28074 1/20 0.34
HRH4 Q9H3N8 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32
HRH1 P35367 1/20 0.32
DGAT1 O75907 1/20 0.31
SOAT1 P35610 1/20 0.31
PIP4K2A P48426 1/20 0.30
PIP4K2C Q8TBX8 1/20 0.30
SSTR4 P31391 1/20 0.30
MBOAT4 Q96T53 1/20 0.30
RXRA P19793 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12240425 0.81 KDM4E (0.40) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL12240466 0.79 KDM4E (0.39) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL21446933 0.78 ADRB3 (0.39) KDM4EPDGFRBPDGFRAPSMB5PIP4K2A
SCHEMBL21367908 0.78 KDM4E (0.38) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL31703760 0.78 KDM4E (0.38) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL16139570 0.78 CHRNB2 (0.41) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL21712544 0.78 KDM4E (0.38) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL595151 0.78 KDM4E (0.38) KDM4EPDGFRBPDGFRAPSMB5
SCHEMBL29911758 0.75 KDM4E (0.39) KDM4EPDGFRBPDGFRAPSMB5HRH4
SCHEMBL23872356 0.75 KDM4E (0.36) KDM4EPDGFRBPDGFRAPSMB5HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021057975-A1 MUTANT IDH2 INHIBITOR AND APPLICATION THEREOF 贝达药业股份有限公司 2021-04-01 WO disclosed