SCHEMBL23196009

SCHEMBL23196009

Cc1cnc(NC(C)(C)C)nc1S(C)(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 2/20 0.41
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CCND2 P30279 1/20 0.38
CCND3 P30281 1/20 0.38
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
AURKA O14965 1/20 0.33
KDR P35968 1/20 0.33
AURKB Q96GD4 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
LRRK2 Q5S007 2/20 0.32
PIM1 P11309 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
MAPK8 P45983 2/20 0.31
MAPK9 P45984 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23196005 0.82 GLP1R (0.40) GLP1RCDK4CCND1CCND2CCND3
SCHEMBL23195819 0.82 GLP1R (0.50) GLP1RCDK4CCND1CCND2CCND3
SCHEMBL23195813 0.78 GLP1R (0.38) GLP1RCDK4CCND1CCND2CCND3
SCHEMBL23196387 0.78 MAPK8 (0.38) GLP1RCDK4CCND1CCND2CCND3
SCHEMBL19145607 0.72 KMT2A (0.33) GLP1RLMNAMAPTKMT2A
SCHEMBL23196358 0.72 GLP1R (0.33) GLP1RCDK4CCND1CCND2CCND3
SCHEMBL270263 0.71 BRD4 (0.52) AURKAJAK2BRD4FLT3
SCHEMBL270248 0.70 JAK1 (0.59) CDK4AURKAKDRAURKBLRRK2
SCHEMBL23196010 0.69 CDK4 (0.36) CDK4CCND1CCND2CCND3AURKA
SCHEMBL21681867 0.65 CDK4 (0.40) CDK4CCND1CCND2CCND3AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4023642-A1 JNK INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF Wuhan LL Science and Technology Development Co., Ltd. (CN) 2022-07-06 EP disclosed
WO-2021063207-A1 JNK INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 武汉朗来科技发展有限公司 2021-04-08 WO disclosed