SCHEMBL23196010

SCHEMBL23196010

CSc1nc(NC(C)(C)C)ncc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
CCND2 P30279 1/20 0.36
CCND3 P30281 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
LRRK2 Q5S007 1/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 1/20 0.33
NPC1 O15118 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
AURKA O14965 1/20 0.32
KDR P35968 1/20 0.32
AURKB Q96GD4 1/20 0.32
PDE4A P27815 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23195815 0.81 SMN1; SMN2 (0.41) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL13734929 0.81 CDK1 (0.38) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL23196386 0.79 MAPK8 (0.39) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL13733999 0.77 KDM4E (0.37) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL13734259 0.74 MAPK8 (0.48) KMT2A
SCHEMBL23196359 0.70
SCHEMBL21711176 0.70 MEN1 (0.34) KMT2ALMNAALDH1A1
SCHEMBL23196009 0.69 GLP1R (0.41) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL21681867 0.68 CDK4 (0.40) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL6181403 0.67 RPS6KA5 (0.34) SMN1; SMN2KMT2AALDH1A1L3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4023642-A1 JNK INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF Wuhan LL Science and Technology Development Co., Ltd. (CN) 2022-07-06 EP disclosed
WO-2021063207-A1 JNK INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 武汉朗来科技发展有限公司 2021-04-08 WO disclosed