SCHEMBL23197829

SCHEMBL23197829

Cc1nc(NC2CCCNC2)nc(C)c1C

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 1/20 0.45
CDK7 P50613 12/20 0.43
CCNH P51946 12/20 0.43
MNAT1 P51948 12/20 0.43
CCNK O75909 9/20 0.43
CDK12 Q9NYV4 9/20 0.43
CCNT1 O60563 8/20 0.43
CDK9 P50750 8/20 0.43
BRD4 O60885 1/20 0.42
PRKCZ Q05513 1/20 0.41
CCNE1 P24864 6/20 0.40
CDK2 P24941 6/20 0.40
MAPK3 P27361 2/20 0.39
MAPK1 P28482 2/20 0.39
SYK P43405 2/20 0.39
KCNH2 Q12809 2/20 0.39
AURKB Q96GD4 2/20 0.39
PLK4 O00444 1/20 0.39
PAK4 O96013 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833890 0.80 IDH2 (0.41) IDH2CDK7CCNHMNAT1CCNK
SCHEMBL25301974 0.80 CCNT1 (0.43) IDH2CDK7CCNHMNAT1CCNK
SCHEMBL25301972 0.80 CCNT1 (0.43) IDH2CDK7CCNHMNAT1CCNK
SCHEMBL23747018 0.77 CCNK (0.58) CDK7CCNHMNAT1CCNKCDK12
SCHEMBL26604076 0.75 IDH2 (0.50) IDH2CDK7CCNHMNAT1CCNK
SCHEMBL26604080 0.75 IDH2 (0.50) IDH2CDK7CCNHMNAT1CCNK
SCHEMBL25596344 0.75 CCNT1 (0.60) CDK7CCNHMNAT1CCNKCDK12
SCHEMBL13524818 0.74 BRD4 (0.52) CDK7CCNHMNAT1CCNKCDK12
SCHEMBL13693348 0.74 BRD4 (0.52) CDK7CCNHMNAT1CCNKCDK12
SCHEMBL31197275 0.74 CCNK (0.44) IDH2CDK7CCNHMNAT1CCNK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021064077-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES AS IRAK4 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2021-04-08 WO disclosed