SCHEMBL23201263

SCHEMBL23201263

CNC(=O)c1ccc2c(=O)[nH]c(=O)[nH]c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.47
IMPDH2 P12268 3/20 0.44
KDM4E B2RXH2 3/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
TTK P33981 1/20 0.43
MAPKAPK2 P49137 1/20 0.42
CSNK2A1 P68400 2/20 0.42
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GAA P10253 1/20 0.41
ITK Q08881 1/20 0.41
SMYD3 Q9H7B4 1/20 0.41
DHODH Q02127 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30882649 1.00 PARP1 (0.47) PARP1IMPDH2KDM4ECA12CA9
SCHEMBL2115397 0.86 XDH (0.47) PARP1IMPDH2KDM4ECA12CA9
SCHEMBL6768125 0.83 SMYD3 (0.55) KDM4EMAPKAPK2ALDH1A1GAASMYD3
SCHEMBL938618 0.81 PARP1 (0.69) PARP1KDM4ECSNK2A1ALDH1A1HPGD
SCHEMBL31042188 0.81 PARP1 (0.69) PARP1KDM4ECSNK2A1ALDH1A1HPGD
SCHEMBL1084591 0.80 PARP1 (0.66) PARP1KDM4ECA12CA9CSNK2A1
SCHEMBL3260502 0.79 PARP1 (0.60) PARP1KDM4ECA12CA9CSNK2A1
SCHEMBL29935457 0.79 PARP1 (0.60) PARP1KDM4ECA12CA9CSNK2A1
SCHEMBL13648691 0.77 PARP1 (0.71) PARP1IMPDH2CSNK2A1CSNK2A2CSNK2B
SCHEMBL14016637 0.77 POLB (0.57) KDM4EMAPKAPK2SMN1; SMN2SMYD3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802489-A2 MASP-2 INHIBITORS AND METHODS OF USE Omeros Corporation (US) 2021-04-14 EP disclosed