Olopatadine

Olopatadine

SCHEMBL23213

CN(C)CC/C=C1/c2ccccc2COc2ccc(CC(=O)O)cc21.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Olopatadine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 3/20 0.98
LMNA P02545 1/20 0.98
PARP1 P09874 1/20 0.77
KDM4E B2RXH2 1/20 0.67
ALDH1A1 P00352 1/20 0.67
RECQL P46063 1/20 0.67
PMP22 Q01453 1/20 0.67
KCNH2 Q12809 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Olopatadine SCHEMBL122589 1.00 HRH1 (0.98) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL29402772 1.00 HRH1 (0.98) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL29381853 1.00 HRH1 (0.98) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL28322959 1.00 HRH1 (0.98) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL2118055 1.00 HRH1 (0.98) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL5324205 1.00 HRH1 (0.98) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL693865 0.99 HRH1 (0.96) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL693866 0.99 HRH1 (0.96) HRH1LMNAPARP1KDM4EALDH1A1
Olopatadine SCHEMBL4669 0.99 HRH1 (1.00) HRH1LMNAPARP1ALDH1A1KCNH2
Olopatadine SCHEMBL29517420 0.99 HRH1 (1.00) HRH1LMNAPARP1ALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4253 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922553-B1 TREATMENT OF ALLERGIC RHINITIS USING A COMBINATION OF MOMETASONE AND OLOPATADINE GLENMARK SPECIALTY SA (CH) 2026-05-06 EP claimed
US-20260076872-A1 POLYMER VIALS WITH SUBSTANTIALLY FLAT BOTTOMS AND INJECTION STRETCH BLOW MOLDING METHODS FOR MAKING THE SAME SIO2 MEDICAL PRODUCTS LLC (US) 2026-03-19 US claimed
CN-121570425-A Olopatadine hydrochloride particles and preparation method thereof 珠海同源药业有限公司 2026-02-27 CN claimed
US-20250242092-A1 SiOx BARRIER FOR PHARMACEUTICAL PACKAGE AND COATING PROCESS SIO2 MEDICAL PRODUCTS INC (US) 2025-07-31 US claimed
US-20250242115-A1 DISPENSING DEVICE AND PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF RHINITIS GLENMARK SPECIALTY S.A. (CH) 2025-07-31 US claimed
EP-4590283-A1 MUCOADHESIVE DRUG DELIVERY SYSTEMS AND METHODS OF USE Madd Ophthalmics Ltd. (CA) 2025-07-30 EP claimed
US-12337065-B2 Compositions for treating viral infections and methods for same ACCESS TO ADVANCED HEALTH INSTITUTE (US) 2025-06-24 US claimed
CN-120189405-A Medical application of olopatadine hydrochloride in treating primary liver cancer diseases 吉林大学 2025-06-24 CN claimed
WO-2025109499-A1 NASAL SPRAY COMPOSITION GLENMARK SPECIALTY S.A. (CH) 2025-05-30 WO claimed
US-20250161328-A1 NASAL SPRAY COMPOSITION GLENMARK SPECIALTY S.A. (CH) 2025-05-22 US claimed
WO-2006051287-A1 COMPOSITION AND METHOD FOR TREATMENT OF ALOPECIA AREATA ARROW INTERNATIONAL LIMITED (MT) 2006-05-18 WO claimed
US-20050256065-A1 Method for stabilizing changes in corneal curvature in an eye by administering compositions containing stabilizing ophthalmic agents PERMASIGHT (US) 2005-11-17 US claimed
EP-1250133-B1 OPHTHALMIC ANTI-ALLERGY COMPOSITIONS SUITABLE FOR USE WITH CONTACT LENSES ALCON INC (CH) 2005-03-30 EP claimed
CN-1483478-A Eye preparation formula adapted for therapentic medicine 无锡杰西医药科技有限公司 2004-03-24 CN claimed
JP-2003520813-A 2003-07-08 JP claimed
EP-1250133-A1 OPHTHALMIC ANTI-ALLERGY COMPOSITIONS SUITABLE FOR USE WITH CONTACT LENSES Alcon Universal, Ltd. (CH) 2002-10-23 EP claimed
US-6375973-B2 OLOPATADINE AND EMEDASTINE AND AN OPHTHALMICALLY ACCEPTABLE POLYMERIC QUATERNARY AMMONIUM COMPOUND AS A PRESERVATIVE ALCON UNIVERSAL LTD. (CH) 2002-04-23 US claimed
US-20010056093-A1 Ophthalmic anti-allergy compositions suitable for use with contact lenses ALCON UNIVERSAL, LTD. 2001-12-27 US claimed
US-20010049369-A1 Brimonidine compositions and methods for retinal degeneration UNIVERSITY OF TENNESSEE RESEARCH CORPORATION, THE 2001-12-06 US claimed
WO-2001054687-A1 OPHTHALMIC ANTI-ALLERGY COMPOSITIONS SUITABLE FOR USE WITH CONTACT LENSES ALCON UNIVERSAL LTD. (CH) 2001-08-02 WO claimed