SCHEMBL23213543

SCHEMBL23213543

Fc1ccc(OCc2ccccc2)c(C2CCN(C3COC4(C3)CN(c3nnco3)C4)CC2)c1.Oc1ccc(F)cc1C1CCN(C2COC3(C2)CN(c2nnco2)C3)CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 9/20 0.48
CHRM1 P11229 9/20 0.48
CHRM2 P08172 3/20 0.38
CHRM5 P08912 1/20 0.38
SLC6A2 P23975 5/20 0.36
SLC6A4 P31645 5/20 0.36
SLC6A3 Q01959 5/20 0.36
HTR1A P08908 4/20 0.36
PTGDR2 Q9Y5Y4 3/20 0.35
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29619684 0.96 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23213891 0.96 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23213887 0.96 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23213301 0.91 CHRM4 (0.47) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23213304 0.89 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5
SCHEMBL23213307 0.89 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5
SCHEMBL23213165 0.87 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23213162 0.87 CHRM4 (0.50) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23230168 0.85 CHRM4 (0.40) CHRM4CHRM1CHRM2CHRM5SLC6A2
SCHEMBL23213875 0.84 CHRM4 (0.53) CHRM4CHRM1CHRM2CHRM5SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021070091-A1 5-OXA-2-AZASPIRO[3.4]OCTANE DERIVATIVES AS M4 AGONISTS NOVARTIS AG (CH) 2021-04-15 WO disclosed