SCHEMBL23217722

SCHEMBL23217722

c1ccc([C@H]2CCc3nc4ccc(-c5cnc(N6CCSCC6)nc5)cc4n32)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TNF P01375 9/20 0.39
EGLN1 Q9GZT9 2/20 0.35
RIPK1 Q13546 3/20 0.33
PTPN11 Q06124 1/20 0.33
AOC3 Q16853 1/20 0.32
CNR2 P34972 1/20 0.31
ACHE P22303 1/20 0.31
NPSR1 Q6W5P4 2/20 0.30
CYP1A2 P05177 1/20 0.30
POLB P06746 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29987401 1.00 TNF (0.39) TNFEGLN1RIPK1PTPN11AOC3
SCHEMBL18151583 0.88 AOC3 (0.43) TNFAOC3CNR2CYP1A2CYP2C9
SCHEMBL18151733 0.88 TNF (0.40) TNFRIPK1AOC3
SCHEMBL29794997 0.88 AOC3 (0.43) TNFAOC3CNR2CYP1A2CYP2C9
SCHEMBL16814754 0.88 AOC3 (0.43) TNFAOC3CNR2CYP1A2CYP2C9
SCHEMBL18151311 0.88 AOC3 (0.43) TNFAOC3CNR2CYP1A2CYP2C9
SCHEMBL29794831 0.87 TNF (0.41) TNFRIPK1AOC3
SCHEMBL18159822 0.87 TNF (0.41) TNFRIPK1AOC3
SCHEMBL18153352 0.86 TNF (0.35) TNFEGLN1PTPN11AOC3
SCHEMBL18150951 0.84 TNF (0.38) TNFRIPK1AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021072269-A1 TARGETED BIFUNCTIONAL DEGRADERS YALE UNIVERSITY (US) 2021-04-15 WO disclosed