SCHEMBL23217766

SCHEMBL23217766

CCOC(=O)Cc1ccccc1OCc1cc(-c2cccc(C(N)C(C)C)c2)c2occc2c1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CFD P00746 19/20 0.59
TPSB2 P20231 8/20 0.47
F11 P03951 7/20 0.47
PTGER1 P34995 1/20 0.38
PTGER4 P35408 1/20 0.38
PTGER3 P43115 1/20 0.38
PTGER2 P43116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30009802 1.00 CFD (0.59) CFDTPSB2F11PTGER1PTGER4
SCHEMBL29095218 0.94 CFD (0.61) CFDTPSB2F11PTGER1PTGER4
SCHEMBL21455658 0.94 CFD (0.61) CFDTPSB2F11PTGER1PTGER4
SCHEMBL29634136 0.94 CFD (0.61) CFDTPSB2F11PTGER1PTGER4
SCHEMBL23656598 0.94 CFD (0.61) CFDTPSB2F11PTGER1PTGER4
SCHEMBL29634229 0.94 CFD (0.61) CFDTPSB2F11PTGER1PTGER4
SCHEMBL23217633 0.91 CFD (0.60) CFDTPSB2F11
SCHEMBL30010133 0.91 CFD (0.60) CFDTPSB2F11
SCHEMBL21455646 0.90 CFD (0.59) CFDTPSB2F11
SCHEMBL29634241 0.90 CFD (0.59) CFDTPSB2F11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4041717-A1 ORAL COMPLEMENT FACTOR D INHIBITORS Biocryst Pharmaceuticals, Inc. (US) 2022-08-17 EP disclosed
CN-114555570-A Oral complement factor D inhibitors 拜奥克里斯特制药公司 2022-05-27 CN disclosed
WO-2021072156-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed
WO-2021072156-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed