SCHEMBL2321984

SCHEMBL2321984

FC(F)(F)c1onc(-c2ccc(Cl)cc2)c1-c1cn(-c2cc[c]cc2)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
FFAR4 Q5NUL3 5/20 0.36
PTGS2 P35354 2/20 0.35
CNR1 P21554 1/20 0.34
PTGS1 P23219 1/20 0.34
PHF8 Q9UPP1 1/20 0.34
MAPT P10636 3/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2318205 0.88 MAP4K4 (0.41) MAP4K4ESR1ESR2FFAR4PTGS2
SCHEMBL2317793 0.87 MAP4K4 (0.39) MAP4K4ESR1ESR2FFAR4PTGS2
SCHEMBL2319332 0.83 MAP4K4 (0.49) MAP4K4ESR1ESR2FFAR4PTGS2
SCHEMBL2320304 0.83 MAPT (0.43) MAP4K4PTGS2PTGS1MAPTALDH1A1
SCHEMBL2318319 0.81 ESR1 (0.52) ESR1ESR2FFAR4PTGS2CNR1
SCHEMBL2318109 0.78 PTGS2 (0.46) ESR1ESR2FFAR4PTGS2MAPT
SCHEMBL2321253 0.77 PTGS2 (0.43) ESR1ESR2FFAR4PTGS2PSEN1
SCHEMBL2317325 0.77 ESR1 (0.48) ESR1ESR2FFAR4PTGS2PTGS1
SCHEMBL2319847 0.77 ESR1 (0.48) ESR1ESR2FFAR4PTGS2PTGS1
SCHEMBL2318956 0.76 ESR1 (0.47) ESR1ESR2FFAR4PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170873-B1 ISOXAZOLE-IMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-08-10 EP disclosed