SCHEMBL2324366

SCHEMBL2324366

[3H]n1ccc(-c2ccccc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
IDO1 P14902 1/20 0.43
METAP2 P50579 1/20 0.43
KEAP1 Q14145 1/20 0.43
RAB9A P51151 2/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
ALOX15 P16050 1/20 0.39
TP53 P04637 1/20 0.37
ALDH1A1 P00352 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35
MAPK1 P28482 1/20 0.35
ASIC3 Q9UHC3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9438 0.76 CYP1A2 (0.48) CYP1A2IDO1METAP2KEAP1RAB9A
SCHEMBL28309054 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
SCHEMBL514705 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
SCHEMBL30636164 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
SCHEMBL31519384 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
Ammonia Solution, Strong SCHEMBL29843017 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
SCHEMBL842040 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
Phosphine SCHEMBL28114703 0.74 CYP1A2 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A
SCHEMBL16800868 0.73 CYP1A2 (0.45) CYP1A2IDO1METAP2KEAP1RAB9A
Bicarbonate SCHEMBL7945138 0.70 TP53 (0.47) CYP1A2IDO1METAP2KEAP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531490-A1 CYCLOHEXYL AMIDE DERIVATIVES AS CRF RECEPTOR ANTAGONISTS Novartis AG (CH) 2012-12-12 EP disclosed
WO-2011095450-A1 CYCLOHEXYL AMIDE DERIVATIVES AS CRF RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2011-08-11 WO disclosed