SCHEMBL23246809

SCHEMBL23246809

Cc1ccc(S(=O)(=O)n2cc(-c3ccc(OC(C)C)c(C#N)c3)c3cc(Br)cnc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.43
XDH P47989 7/20 0.41
S1PR1 P21453 5/20 0.38
S1PR5 Q9H228 3/20 0.38
RORC P51449 1/20 0.36
TBK1 Q9UHD2 1/20 0.36
S1PR3 Q99500 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31396624 1.00 PTPN11 (0.43) PTPN11XDHS1PR1S1PR5RORC
SCHEMBL31396554 0.91 PTPN11 (0.45) PTPN11XDH
SCHEMBL23248021 0.88 PTPN11 (0.43) PTPN11XDHS1PR1S1PR5RORC
SCHEMBL15607356 0.87 PTPN11 (0.42) PTPN11XDHS1PR1TBK1
SCHEMBL15607353 0.83 TBK1 (0.49) TBK1
SCHEMBL15607501 0.83 TBK1 (0.41) PTPN11TBK1
SCHEMBL31396556 0.82 PTPN11 (0.47) PTPN11KCNH2
SCHEMBL15607458 0.82 TBK1 (0.44) PTPN11TBK1
SCHEMBL31396616 0.81 PTPN11 (0.53) PTPN11
SCHEMBL15554915 0.81 PTPN11 (0.43) PTPN11XDHTBK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021074279-A1 SPIRO-FUSED TRICYCLIC MAP4K1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2021-04-22 WO disclosed