SCHEMBL23247129

SCHEMBL23247129

Nc1ccc(N2C[C@H]3C[C@@H]2CN3C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.47
FAAH O00519 1/20 0.38
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
HDAC1 Q13547 2/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
CASP6 P55212 1/20 0.34
GFER P55789 1/20 0.34
MAP3K12 Q12852 1/20 0.33
RORC P51449 2/20 0.33
BRAF P15056 1/20 0.33
BTK Q06187 2/20 0.33
CYP2C8 P10632 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23247188 1.00 AKR1C3 (0.47) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL4668901 0.86 AKR1C3 (0.48) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL30307832 0.86 AKR1C3 (0.48) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL4668904 0.86 AKR1C3 (0.48) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL4668899 0.86 AKR1C3 (0.48) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL23538793 0.86 AKR1C3 (0.48) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL2723382 0.82 CHRNB2 (0.56) AKR1C3FAAHHDAC1CHRNB2CHRNA4
SCHEMBL16872560 0.82 CHRNB2 (0.56) AKR1C3FAAHHDAC1CHRNB2CHRNA4
SCHEMBL1017691 0.82 AKR1C3 (0.45) AKR1C3FAAHDRD2DRD4DRD3
SCHEMBL23247148 0.80 AKR1C3 (0.43) AKR1C3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021074251-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER SENTINEL ONCOLOGY LIMITED (GB) 2021-04-22 WO disclosed