SCHEMBL23264274

SCHEMBL23264274

O=C(Nc1c(Br)cc(C(F)(C(F)(F)F)C(F)(F)F)cc1OC(F)F)c1cccc(N(CC2CC2)C(=O)c2ccc(F)cc2)c1F

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 11/20 0.35
PDE4D Q08499 8/20 0.35
PDE4A P27815 6/20 0.35
PDE4C Q08493 6/20 0.35
ABCB11 O95342 1/20 0.35
HDAC8 Q9BY41 2/20 0.34
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
AR P10275 1/20 0.30
S1PR1 P21453 1/20 0.30
SCN8A Q9UQD0 1/20 0.30
SCN10A Q9Y5Y9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29431922 1.00 PDE4B (0.35) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264310 0.95 PDE4B (0.35) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264279 0.95 PDE4B (0.34) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL29431906 0.95 PDE4B (0.34) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264314 0.94 PDE4B (0.38) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264311 0.92 PDE4B (0.35) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264315 0.91 PDE4B (0.32) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264286 0.91 PDE4B (0.38) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL29431915 0.91 PDE4B (0.38) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL23264313 0.91 DHODH (0.34) PDE4BPDE4DPDE4APDE4CABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112707841-B 3-N-cyclopropylmethyl-2-fluorobenzamide compound and preparation method and application thereof 南通泰禾化工股份有限公司 2022-08-23 CN disclosed
CN-112661665-B Amide compound and preparation method and application thereof 南通泰禾化工股份有限公司 2021-09-14 CN disclosed
WO-2021078293-A1 3-N-CYCLOPROPYLMETHYL-2-FLUOROBENZAMIDE COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 南通泰禾化工股份有限公司 2021-04-29 WO disclosed
CN-112707841-A 3-N-cyclopropylmethyl-2-fluorobenzamide compound and preparation method and application thereof 南通泰禾化工股份有限公司 2021-04-27 CN disclosed
WO-2021073373-A1 AMIDE COMPOUNDS AND PREPARATION METHOD THEREFOR AND USE THEREOF CAC NANTONG CHEMICAL CO., LTD. (CN) 2021-04-22 WO disclosed
CN-112661665-A Amide compound and preparation method and application thereof 南通泰禾化工股份有限公司 2021-04-16 CN disclosed