SCHEMBL23267271

SCHEMBL23267271

O=C1CCC(N2Cc3cc(C#CSI)ccc3C2=O)C(=O)N1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 10/20 0.64
IKZF2 Q9UKS7 10/20 0.52
CSNK1A1 P48729 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24637376 0.87 CRBN (0.69) CRBNIKZF2CSNK1A1
SCHEMBL30569130 0.87 CRBN (0.69) CRBNIKZF2CSNK1A1
SCHEMBL21877059 0.85 CRBN (0.64) CRBNIKZF2CSNK1A1
SCHEMBL29488410 0.84 CRBN (0.69) CRBNIKZF2CSNK1A1
SCHEMBL21760044 0.84 CRBN (0.69) CRBNIKZF2CSNK1A1
SCHEMBL24601235 0.84 CRBN (0.69) CRBNIKZF2CSNK1A1
SCHEMBL1413817 0.84 CRBN (0.69) CRBNIKZF2CSNK1A1
SCHEMBL23250036 0.84 CRBN (0.62) CRBNIKZF2CSNK1A1
SCHEMBL21759818 0.84 CRBN (0.65) CRBNIKZF2CSNK1A1
SCHEMBL20129297 0.84 CRBN (0.62) CRBNIKZF2CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021077010-A1 BIFUNCTIONAL MOLECULES CONTAINING AN E3 UBIQUITINE LIGASE BINDING MOIETY LINKED TO A BCL6 TARGETING MOIETY ARVINAS OPERATIONS, INC. (US) 2021-04-22 WO disclosed