SCHEMBL23315467

SCHEMBL23315467

CCOC(=O)C1Cc2c(ccc(OC)c2OCc2ccc(OC)cc2)CN1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 12/20 0.49
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
AGTR1 P30556 2/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21881614 1.00 AGTR2 (0.49) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL21881186 0.91 AGTR2 (0.49) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL21881194 0.91 AGTR2 (0.49) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL21881185 0.91 AGTR2 (0.59) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL18608232 0.91 AGTR2 (0.59) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL21881848 0.91 AGTR2 (0.59) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL29758892 0.90 AGTR2 (0.58) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL21596260 0.90 AGTR2 (0.58) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL21881369 0.89 AGTR2 (0.49) AGTR2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL21881515 0.89 AGTR2 (0.47) AGTR2KDM4ECYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3620454-B1 CARBOXYLIC ACID DERIVATIVE AS AT2R RECEPTOR ANTAGONIST SHANDONG DANHONG PHARMACEUTICAL CO LTD (CN) 2021-05-05 EP disclosed