SCHEMBL23316631

SCHEMBL23316631

Bc1c(O)c(O)c(O)c(/C(O)=c2\[nH]c(=O)/c(=C(\O)c3nc[nH]c3C(C)(C)C)[nH]c2=O)c1O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.33
CYP1A2 P05177 1/20 0.33
CDK1 P06493 1/20 0.33
CYP2C9 P11712 1/20 0.33
CCNB1 P14635 1/20 0.33
CYP2C19 P33261 1/20 0.33
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32
TUBB2A Q13885 1/20 0.32
TUBB8 Q3ZCM7 1/20 0.32
TUBA3E Q6PEY2 1/20 0.32
TUBA1A Q71U36 1/20 0.32
TUBA1C Q9BQE3 1/20 0.32
TUBB6 Q9BUF5 1/20 0.32
TUBB2B Q9BVA1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20081578 0.94 RAF1 (0.33) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL23316771 0.82 CYP1A2 (0.46) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL20081366 0.81 CYP1A2 (0.55) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL23316809 0.78 CYP1A2 (0.55) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL20081635 0.77 CYP1A2 (0.47) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL20081584 0.74 CYP1A2 (0.41) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL20081625 0.72 RAF1 (0.33) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL20177151 0.67 CYP1A2 (0.44) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL20177153 0.67 TUBB4A (0.46) RAF1CYP1A2CDK1CYP2C9CCNB1
SCHEMBL24444426 0.66 CYP1A2 (0.43) RAF1CYP1A2CDK1CYP2C9CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3312163-B1 DEUTERIUM-SUBSTITUTED DEHYDROPHENYLAHISTIN-LIKE COMPOUNDS, PREPARATION METHOD THEREOF AND USE IN PREPARATION OF ANTITUMOR DRUG MARINE BIOMEDICAL RES INST QINGDAO CO LTD (CN) 2021-05-05 EP disclosed